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Screening
Affinity determination
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Chemistry Methods
2024
4 (10)
Article · Drug discovery
Rescaling NMR for a Larger Deployment in Drug Discovery: Hyperpolarization and Benchtop NMR as Potential Game-Changers
M. Bütikofer, G. R. Stadler, F. Torres
Chemistry Methods 2024, 4, e202400009
JACS
2024
146 (26)
Article · Drug discovery · Affinity determination
Rapid Protein–Ligand Affinity Determination by Photoinduced Hyperpolarized NMR
M. Bütikofer, G. R. Stadler, H. Kadavath, R. Cadalbert, F. Torres, R. Riek
J. Am. Chem. Soc. 2024, 146, 17974–17985
Magritek
2024
Application note · Drug discovery
Let your NMR signal shine – Automated photoCIDNP experiments with a Spinsolve benchtop NMR
Magritek, 1 March 2024
JACS
2023
145 (22)
Article · Drug discovery · Screening
Ultrafast Fragment Screening Using Photo-Hyperpolarized (CIDNP) NMR
F. Torres, M. Bütikofer, G. R. Stadler, A. Renn, H. Kadavath, R. Bobrovs, K. Jaudzems, R. Riek
J. Am. Chem. Soc. 2023, 145, 12066–12080